SCHEMBL17629909

SCHEMBL17629909

Cc1cc(C#N)ccc1-c1ccc(Br)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
S1PR1 P21453 1/20 0.42
EGLN2 Q96KS0 6/20 0.42
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41
CYP11B2 P19099 6/20 0.41
CYP11B1 P15538 5/20 0.41
KDM1A O60341 1/20 0.38
AHR P35869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17630042 0.89 MAOB (0.43) MAOAMAOBS1PR1CYP11B2CYP11B1
SCHEMBL7634772 0.89 ALDH1A1 (0.48) S1PR1EGLN2PDE3BPDE3AHRH2
SCHEMBL27806613 0.87 KIF11 (0.47) S1PR1EGLN2PDE3BPDE3AHRH2
SCHEMBL23625527 0.85 ALDH1A1 (0.56) S1PR1EGLN2PDE3BPDE3AHRH2
SCHEMBL12496569 0.82 PTGS1 (0.49) S1PR1EGLN2PDE3BPDE3AHRH2
SCHEMBL2786090 0.82 MMP3 (0.57) MAOAEGLN2HRH2HRH1CYP11B2
SCHEMBL2572264 0.81 ESR2 (0.53) EGLN2CYP11B2CYP11B1
SCHEMBL2154193 0.80 CYP11B2 (0.53) EGLN2PDE3BPDE3ACYP11B2CYP11B1
SCHEMBL25767772 0.80 CYP11B1 (0.45) S1PR1EGLN2PDE3BPDE3AHRH2
SCHEMBL7229011 0.79 HRH2 (0.47) MAOAMAOBHRH2HRH1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016046782-A1 IMIDAZOLE BIARYL COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-03-31 WO disclosed