SCHEMBL17635528

SCHEMBL17635528

CC(=O)c1cc(N)cc(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.43
CREBBP Q92793 1/20 0.41
NPC1 O15118 3/20 0.38
MAPT P10636 3/20 0.38
RAB9A P51151 1/20 0.38
PARP1 P09874 1/20 0.36
MTOR P42345 1/20 0.36
LMNA P02545 1/20 0.36
PRKCI P41743 1/20 0.36
FURIN P09958 1/20 0.35
KDM4E B2RXH2 2/20 0.34
NOTUM Q6P988 1/20 0.33
MAOB P27338 3/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
MAOA P21397 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1976289 0.84 CA5A (0.52) CA5ACREBBPNPC1MAPTRAB9A
SCHEMBL2628599 0.84 CA5A (0.52) CA5ACREBBPNPC1MAPTRAB9A
SCHEMBL15709749 0.84 CA5A (0.52) CA5ANPC1MAPTRAB9APARP1
SCHEMBL343284 0.84 CA5A (0.52) CA5ANPC1MAPTRAB9APARP1
SCHEMBL7184528 0.82 PBRM1 (0.42) NPC1MAPTRAB9APARP1LMNA
SCHEMBL30197207 0.80 KDM4E (0.47) CA5AMAPTPARP1LMNAKDM4E
SCHEMBL1028516 0.80 KDM4E (0.47) CA5AMAPTPARP1LMNAKDM4E
SCHEMBL15484864 0.80 PARP1 (0.52) MAPTPARP1LMNAKDM4EHTT
SCHEMBL24150559 0.78 TUBB4A (0.46) CREBBPMTORLMNAKDM4EHTT
SCHEMBL176618 0.78 NOTUM (0.57) NPC1MAPTLMNAKDM4ENOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597087-B1 Dihydrooxazine and tetrahydropyrimidine derivatives as BACE 1 inhibitors SHIONOGI & CO (JP) 2016-03-30 EP disclosed