SCHEMBL1778129

SCHEMBL1778129

CC(C)(NC(=O)c1cc2c(NC(=O)c3ccccc3NC(=O)c3ccccc3F)n[nH]c2s1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.43
PPARG P37231 3/20 0.42
NR1H4 Q96RI1 2/20 0.42
ABL1 P00519 2/20 0.41
BCR P11274 2/20 0.41
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
IMPDH2 P12268 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
ALDH1A1 P00352 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
FGFR4 P22455 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 1/20 0.36
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741093 0.96 AURKA (0.46) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1779700 0.91 AURKA (0.50) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1778008 0.91 AURKA (0.49) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1779328 0.90 RXFP1 (0.44) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1780795 0.90 AURKA (0.45) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1779010 0.88 RXFP1 (0.48) AURKAABL1BCRNPC1RAB9A
SCHEMBL1780888 0.88 RXFP1 (0.46) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1780912 0.88 AURKA (0.49) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1779573 0.88 AURKA (0.43) AURKAPPARGNR1H4ABL1BCR
SCHEMBL1779104 0.87 AURKA (0.43) AURKAPPARGNR1H4ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943654-B2 1H-thieno[2,3-c]pyrazole compounds useful as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2011-05-17 US disclosed