SCHEMBL17801014

SCHEMBL17801014

Brc1n[nH]c2ccc(-c3ncc[nH]3)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.47
MTOR P42345 1/20 0.46
ADK P55263 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MAP3K8 P41279 1/20 0.42
TLR9 Q9NR96 1/20 0.41
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
JAK2 O60674 5/20 0.39
CDK2 P24941 2/20 0.39
DCLK1 O15075 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377574 0.79 CSNK1D (0.46) NISCHPDE3BPDE3AALDH1A1MAP3K8
SCHEMBL17801023 0.76 LRRK2 (0.52) MAP3K8MKNK1CHEK1
SCHEMBL722191 0.74 NISCH (0.78) NISCHMTORADKPDE3BPDE3A
SCHEMBL17801062 0.74 BTK (0.50) JAK2CDK2DCLK1PRKD3MAP4K4
SCHEMBL8253395 0.73 VCP (0.47) NISCHMTORADKJAK2MKNK1
SCHEMBL482406 0.73 NISCH (0.64) NISCHMTORADKPDE3BPDE3A
SCHEMBL17801017 0.72 PDPK1 (0.60) KDM4EALDH1A1CHEK1PDPK1
SCHEMBL17801025 0.72 LRRK2 (0.50) CLK4MKNK1PDPK1
SCHEMBL862114 0.72 NISCH (0.75) NISCHMTORADKPDE3BPDE3A
SCHEMBL5914856 0.71 NISCH (0.62) NISCHMTORADKPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed