SCHEMBL17801241

SCHEMBL17801241

Cc1nc(C(=O)O)cc2sc(NC(C)C)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
ALOX15 P16050 2/20 0.38
HSD17B10 Q99714 2/20 0.38
PKM P14618 1/20 0.38
KDM4E B2RXH2 2/20 0.36
PTP4A3 O75365 1/20 0.36
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
CDK5 Q00535 2/20 0.34
CDK5R1 Q15078 2/20 0.34
NPC1 O15118 2/20 0.34
HTT P42858 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
TP53 P04637 1/20 0.34
GSK3A P49840 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695319 0.75 MAPK14 (0.42) CCNA2CDK2MAPTKDM4EPTP4A3
SCHEMBL1180045 0.68 MAPK1 (0.47) ALDH1A1MAPTALOX15KDM4EGAA
SCHEMBL23628970 0.68 SMN1; SMN2 (0.54) ALDH1A1MAPTHSD17B10KDM4EGAA
SCHEMBL21062055 0.67 HCAR3 (0.46) CCNA2CDK2ALDH1A1MAPTALOX15
SCHEMBL8142798 0.66 CDK2 (0.42) CCNA2CDK2ALDH1A1MAPTALOX15
SCHEMBL2744060 0.66 L3MBTL1 (0.62) CCNA2CDK2ALDH1A1MAPTKDM4E
SCHEMBL17801297 0.65 CYP1A2 (0.52) ALDH1A1MAPTKDM4ENPC1HTT
Bromide SCHEMBL2241396 0.65 L3MBTL1 (0.60) CCNA2CDK2ALDH1A1MAPTKDM4E
SCHEMBL1425069 0.65 ALOX15 (0.38) ALDH1A1MAPTALOX15KDM4ESMN1; SMN2
SCHEMBL18358191 0.65 KDM4E (0.49) MAPTALOX15KDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227301-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2017-10-11 EP disclosed
EP-2266981-B1 Benzothiazole compounds useful as kinase inhibitors BRISTOL MYERS SQUIBB CO (US) 2016-07-06 EP disclosed
WO-2016087417-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed