SCHEMBL17814737

SCHEMBL17814737

Nc1c(N=O)c(=O)nc(S)n1Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPK10 P53779 1/20 0.41
TNF P01375 1/20 0.39
CXCL8 P10145 1/20 0.39
SOS1 Q07889 1/20 0.39
NOD2 Q9HC29 1/20 0.39
NOD1 Q9Y239 1/20 0.39
KDM4E B2RXH2 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TYMS P04818 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814738 0.83 TNF (0.42) ALDH1A1TNFCXCL8SOS1NOD2
SCHEMBL28538573 0.79 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28547235 0.76 RAB9A (0.45) ALDH1A1CYP1A2CYP3A4CYP2C19TNF
SCHEMBL7674391 0.72 MEN1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL29172412 0.72 P2RX3 (0.41) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28551647 0.72
SCHEMBL17814735 0.69 PNP (0.57) KMT2ATLR7TLR8
SCHEMBL28537635 0.69 TSHR (0.37) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3239986 0.68 NPSR1 (0.52) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4181999 0.68 SMN1; SMN2 (0.40) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed
WO-2016088838-A1 PURINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF 塩野義製薬株式会社 2016-06-09 WO disclosed