SCHEMBL17844150

SCHEMBL17844150

CC(C)(C)n1sc(-c2ccccc2)c(NCCc2ccccn2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.45
CYP1A2 P05177 2/20 0.42
MAOB P27338 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
CASP3 P42574 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TAAR1 Q96RJ0 1/20 0.40
ALOX15 P16050 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
HIF1A Q16665 1/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
APP P05067 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CYP2C19 P33261 1/20 0.37
AURKA O14965 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844176 0.82 ADORA3 (0.35) ADORA1AURKA
SCHEMBL17844227 0.78 POLB (0.39) LMNAALDH1A1HTTSMN1; SMN2AURKA
SCHEMBL3551960 0.76 BRD4 (0.39) ALDH1A1SMN1; SMN2
SCHEMBL5261593 0.74 MAPT (0.40) CYP1A2LMNAALDH1A1TAAR1TDP1
SCHEMBL17844148 0.73 KMT2A (0.40) ALDH1A1TDP1RAB9ANPC1HTT
SCHEMBL17844175 0.73 CA12 (0.38) ALDH1A1CYP2C19
SCHEMBL17844195 0.71 ASPH (0.41) MKNK1MAOBALDH1A1ALOX15TDP1
SCHEMBL17844088 0.71 KDM4E (0.40) CYP1A2LMNAALDH1A1ALOX15TDP1
SCHEMBL2002898 0.68 NR1H2 (0.47) MKNK1CYP1A2MAOBHRH3LMNA
SCHEMBL28731705 0.65 CYP1A2 (0.60) CYP1A2HRH3LMNAALDH1A1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed