SCHEMBL17844873

SCHEMBL17844873

CC(C)(C)OC(=O)C(N)(CCCCc1ccccc1)OS(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.40
GRM3 Q14832 1/20 0.40
NAAA Q02083 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PTPRC P08575 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPRB P23467 1/20 0.39
PTPRG P23470 1/20 0.39
ACP1 P24666 1/20 0.39
LTB4R Q15722 4/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844787 0.96 PTPRC (0.42) GRM2GRM3NAAAMMP1MMP2
SCHEMBL17844847 0.83 CA12 (0.43) MMP1PTPN2PTPN1PTPRBCA12
SCHEMBL9296370 0.78 GRM2 (0.47) GRM2GRM3NAAALTB4RPOLB
SCHEMBL7445828 0.76 LTB4R (0.44) GRM2GRM3NAAALTB4RPOLB
SCHEMBL9414314 0.75 KDM4E (0.40) LMNA
SCHEMBL8315125 0.74 SMN1; SMN2 (0.46) GRM2GRM3PTPRCPTPN2PTPN1
SCHEMBL7034400 0.71 DGAT1 (0.34) CA12CA1CA7CA14
SCHEMBL7283510 0.71 FAAH (0.45) PTPRCPTPN2PTPN1PTPRBPTPRG
SCHEMBL9543962 0.71 SMN1; SMN2 (0.49) GRM2GRM3CA12CA1CA7
SCHEMBL4385270 0.71 SMN1; SMN2 (0.49) GRM2GRM3CA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095088-A1 ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed