SCHEMBL17848759

SCHEMBL17848759

CC(C)(C)OC(=O)N1CCC2(CC1)CCN2c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 3/20 0.56
ATM Q13315 1/20 0.52
CCR5 P51681 2/20 0.50
USP30 Q70CQ3 1/20 0.50
TSHR P16473 2/20 0.49
ALOX15 P16050 1/20 0.49
NPC1L1 Q9UHC9 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
MEN1 O00255 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
USP2 O75604 2/20 0.46
HSD17B10 Q99714 1/20 0.46
TACR1 P25103 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17777790 0.87 GPR119 (0.50) GPR119ATMCCR5USP30TSHR
SCHEMBL38661929 0.86 HIF1A (0.49) GPR119ATMTSHRCYP3A4CYP2C19
SCHEMBL20212767 0.86 MEN1 (0.54) GPR119MEN1KMT2AUSP2HSD17B10
SCHEMBL745368 0.84 GPR119 (0.51) GPR119ATMCCR5USP30TSHR
SCHEMBL17848630 0.81 MEN1 (0.54) GPR119MEN1KMT2AUSP2HSD17B10
SCHEMBL5095029 0.80 GPR119 (0.50) GPR119ATMCCR5USP30TSHR
SCHEMBL17140706 0.79 GPR119 (0.49) GPR119ATMCCR5USP30TSHR
SCHEMBL318858 0.79 CCR5 (0.75) GPR119CCR5HSD17B10OPRD1OPRK1
SCHEMBL7845129 0.79 NPC1L1 (0.58) GPR119ATMCCR5USP30NPC1L1
SCHEMBL17140692 0.79 NPC1L1 (0.58) GPR119ATMCCR5USP30NPC1L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-B1 DOPAMINE D2 RECEPTOR LIGANDS BROAD INST INC (US) 2026-05-06 EP disclosed
US-12428373-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2025-09-30 US disclosed
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
US-11498896-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2022-11-15 US disclosed
US-20210147355-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2021-05-20 US disclosed
US-10633336-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2020-04-28 US disclosed
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2018-06-07 US disclosed
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2018-06-07 US disclosed
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, DRD3, ARRB1 GPR119 73/4885ATM 2909/4885CCR5 320/4885
US-11498896-B2 Dopamine D2 receptor ligands DRD2, SLC6A3, NTSR2 GPR119 134/4885ATM 4111/4885CCR5 626/4885
US-10633336-B2 Dopamine D2 receptor ligands DRD2, ARRB1, DRD3 GPR119 145/4885ATM 2761/4885CCR5 353/4885
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 GPR119 134/4885ATM 4111/4885CCR5 626/4885
US-20210147355-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 GPR119 134/4885ATM 4111/4885CCR5 626/4885
US-12428373-B2 Dopamine D2 receptor ligands DRD2, SLC6A3, NTSR2 GPR119 134/4885ATM 4111/4885CCR5 626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.