SCHEMBL17849206

SCHEMBL17849206

N=C(c1ccc(OCC(=O)NCCO)cc1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ACACA Q13085 1/20 0.35
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
PDK2 Q15119 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
GAA P10253 1/20 0.33
ALOX12 P18054 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623547 0.87 SYK (0.36) ALDH1A1KDM4ETDP1
SCHEMBL16726696 0.86 HDAC6 (0.41) ALDH1A1RAB9ASMN1; SMN2KDM4EHTT
SCHEMBL17849220 0.82 MT-CO2 (0.35) KDM4E
SCHEMBL16623588 0.81 SYK (0.34)
SCHEMBL16726674 0.78 PRKAB2 (0.35)
SCHEMBL16726665 0.77 ALDH2 (0.33) KMT2A
SCHEMBL16623450 0.74 NPC1 (0.32) HTT
SCHEMBL17849208 0.73 HDAC6 (0.33) ALDH1A1KMT2ASMN1; SMN2
SCHEMBL17849205 0.72 DGAT1 (0.32) ALDH1A1
SCHEMBL17849236 0.72 RORC (0.36) KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed