SCHEMBL17850259

SCHEMBL17850259

NNC(=O)c1cc(O)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.50
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 3/20 0.47
GFER P55789 2/20 0.47
MPO P05164 2/20 0.44
CYP3A4 P08684 2/20 0.44
BLM P54132 2/20 0.44
KDM5A P29375 1/20 0.44
PMP22 Q01453 1/20 0.44
HIF1A Q16665 1/20 0.44
CYP1A2 P05177 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C19 P33261 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
ANO1 Q5XXA6 3/20 0.39
SMYD3 Q9H7B4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7171815 0.81 KDM4E (0.57) P2RX7ALDH1A1KDM4EGFERMPO
SCHEMBL30201887 0.81 KDR (0.47) ALDH1A1KDM4ECYP3A4PMP22CYP1A2
SCHEMBL27212647 0.81 P2RX7 (0.50) P2RX7ALDH1A1KDM4EMPOCYP3A4
SCHEMBL3257638 0.81 KDR (0.47) ALDH1A1KDM4ECYP3A4PMP22CYP1A2
SCHEMBL31345733 0.81 P2RX7 (0.50) P2RX7ALDH1A1KDM4EMPOCYP3A4
SCHEMBL31213280 0.79 P2RX7 (0.49) P2RX7KDM4EMPOCYP3A4CYP1A2
SCHEMBL1505656 0.79 ALDH1A1 (0.61) P2RX7ALDH1A1KDM4EMPOCYP3A4
SCHEMBL107759 0.79 CTSA (0.50) P2RX7KDM4E
SCHEMBL29679606 0.79 ALDH1A1 (0.61) P2RX7ALDH1A1KDM4EMPOCYP3A4
SCHEMBL1054692 0.79 KDM4C (0.58) P2RX7ALDH1A1KDM4ECYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240317978-A1 RUBBER COMPOSITION AND TIRE OTSUKA CHEMICAL CO., LTD. (JP) 2024-09-26 US disclosed
EP-4365229-A1 RUBBER COMPOSITION AND TIRE Otsuka Chemical Co., Ltd. (JP) 2024-05-08 EP disclosed
CN-117561303-A Rubber composition and tire 大塚化学株式会社 2024-02-13 CN disclosed
EP-2424869-B1 5,6,7,8-TETRAHYDRO[1,2,4]TRIAZOLO[4,3-a]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LTD (GB) 2016-06-22 EP disclosed