SCHEMBL17853274

SCHEMBL17853274

Cn1ncc(NC(=O)OP)c1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
BPTF Q12830 1/20 0.33
KAT2B Q92831 2/20 0.33
BRD9 Q9H8M2 1/20 0.33
ALDH1A1 P00352 3/20 0.32
HTT P42858 3/20 0.32
KDM4E B2RXH2 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 1/20 0.31
LPAR1 Q92633 1/20 0.31
PIM1 P11309 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
PKM P14618 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5497757 0.80 BRD9 (0.36) CNR2CYP1A2CYP2C19BPTFKAT2B
SCHEMBL3114686 0.78 ALDH1A1 (0.46) CYP1A2ALDH1A1HTTKDM4EMEN1
SCHEMBL16592882 0.73 KAT2B (0.33) CNR2CYP1A2CYP2C19BPTFKAT2B
SCHEMBL3120670 0.72 PKM (0.47) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL5500017 0.71 TLR7 (0.36) ALDH1A1KDM4EHDAC1
SCHEMBL16592911 0.71 GLA (0.34) CNR2CYP1A2CYP2C19ALDH1A1HTT
SCHEMBL15856849 0.71 NTRK1 (0.37) BPTFKAT2BBRD9MEN1KMT2A
SCHEMBL6065170 0.71 HTT (0.47) ALDH1A1HTTKDM4EMEN1KMT2A
SCHEMBL16078095 0.71 L3MBTL1 (0.44) CYP1A2CYP2C19KDM4EHDAC1HDAC2
SCHEMBL5493771 0.70 CCNC (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095860-A1 PYRAZOLYL CARBOXYLIC ACID AND PYRAZOLYL UREA DERIVATIVE COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed