SCHEMBL17866019

SCHEMBL17866019

[CH2][C@H]1C[C@@H](n2cc(F)c3c(NCc4ccccc4)ncnc32)C[C@@H]1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 2/20 0.46
SIGMAR1 Q99720 2/20 0.45
ADRA2C P18825 1/20 0.45
OPRK1 P41145 1/20 0.45
HTR2B P41595 1/20 0.45
HTR6 P50406 1/20 0.45
PDE11A Q9HCR9 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
TP53 P04637 2/20 0.41
ABL1 P00519 1/20 0.40
EGFR P00533 1/20 0.40
ABL2 P42684 1/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 1/20 0.40
MAPK10 P53779 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADORA3 P0DMS8 5/20 0.39
SLC29A1 Q99808 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADORA2A P29274 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865954 0.83 ADK (0.46) ADKSIGMAR1ADRA2COPRK1HTR2B
SCHEMBL12986946 0.81 NAE1 (0.59)
SCHEMBL191643 0.81 NAE1 (0.59)
SCHEMBL17875173 0.79 SIGMAR1 (0.42) ADKSIGMAR1ADRA2COPRK1HTR2B
SCHEMBL5465354 0.73 NAE1 (0.41) ADKABL1EGFRABL2LCK
SCHEMBL12983619 0.73 POLB (0.43) ADKADORA3ADORA2AADORA1
SCHEMBL10236879 0.73 NAE1 (0.43) ADKSIGMAR1ADRA2COPRK1HTR2B
SCHEMBL17866056 0.72 TP53 (0.47) SIGMAR1HTR2BTP53ABL1EGFR
SCHEMBL17866039 0.72 UBA6 (0.44) EGFR
SCHEMBL10005047 0.71 ADORA3 (0.52) ADORA3SLC29A1ADORA2AADORA1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402334-B1 Inhibitors of E1 Activating Enzymes MILLENNIUM PHARM INC (US) 2016-06-29 EP claimed