SCHEMBL17870951

SCHEMBL17870951

C#Cc1cccc(N2CCC2=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GAA P10253 1/20 0.40
NSD2 O96028 1/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
LMNA P02545 1/20 0.39
ALOX5 P09917 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23120599 0.81 CRBN (0.64) ALDH1A1HPGDNSD2DDB1CRBN
SCHEMBL2518608 0.75 ALDH1A1 (0.59) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL15273560 0.75 DDB1 (0.65) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL3551042 0.74 ALOX5 (0.59) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL9564052 0.74 L3MBTL1 (0.62) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL9407810 0.74 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL17870929 0.74 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL4411364 0.73 ALOX5 (0.55) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL3936113 0.73 NSD2 (0.74) ALDH1A1GAANSD2LMNASMN1; SMN2
SCHEMBL30516650 0.72 ALOX5 (0.55) ALDH1A1CYP3A4CYP2C9CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3224245-A1 NECROSIS INHIBITORS National Institute Of Biological Sciences, Beijing (CN) 2017-10-04 EP disclosed
WO-2016101887-A1 NECROSIS INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2016-06-30 WO disclosed