SCHEMBL17892183

SCHEMBL17892183

CC(C)C(CNC(=O)O)c1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
KCNA3 P22001 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
CYP1A2 P05177 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
CTSK P43235 2/20 0.41
CNR1 P21554 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALOX5 P09917 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2549352 0.83 CYP1A2 (0.46) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL1554808 0.77 BCAT2 (0.51) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL17373696 0.77 BCAT2 (0.51) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL17892155 0.77 SLC6A2 (0.60) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL17892157 0.77 SLC6A2 (0.60) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL19692700 0.76 CNR1 (0.42) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL2553821 0.74 P4HB (0.42) KCNA3
Bromobenzene SCHEMBL27905968 0.74 CYP2C19 (0.63) SMN1; SMN2CYP1A2ALDH1A1LMNACYP2D6
SCHEMBL3655014 0.72 MTNR1A (0.58) SMN1; SMN2SLC6A4ALDH1A1LMNACYP2D6
SCHEMBL3655009 0.72 MTNR1A (0.58) SMN1; SMN2SLC6A4ALDH1A1LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109501-A1 AMIDE COMPOUNDS AS TRYPTOPHAN HYDROXYLASE INHIBITORS KAROS PHARMACEUTICALS, INC. (US) 2016-07-07 WO disclosed