SCHEMBL10175449

SCHEMBL10175449

Cn1c(-c2ccncc2Br)nc2ccc(F)c(F)c21

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.60
CYP11B1 P15538 4/20 0.36
PDE10A Q9Y233 6/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ATM Q13315 1/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
PDE2A O00408 4/20 0.32
NOS2 P35228 2/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
PDE7A Q13946 1/20 0.31
LATS1 O95835 1/20 0.30
LATS2 Q9NRM7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175451 0.86 CYP11B2 (0.63) CYP11B2CYP11B1PDE10APOLBSMN1; SMN2
SCHEMBL463351 0.84 CYP11B2 (0.67) CYP11B2CYP11B1PDE10APDE2ANOS2
SCHEMBL10175454 0.83 CYP11B2 (0.53) CYP11B2CYP11B1
SCHEMBL10175118 0.81 CYP11B2 (0.57) CYP11B2CYP11B1PDE10APOLBSMN1; SMN2
SCHEMBL17896706 0.80 CYP11B2 (0.61) CYP11B2CYP11B1PDE10APOLBSMN1; SMN2
SCHEMBL17896708 0.77 CYP11B2 (0.68) CYP11B2CYP11B1
SCHEMBL10175447 0.76 CYP11B2 (0.60) CYP11B2CYP11B1ATMDPP4DPP8
SCHEMBL10175463 0.76 CYP11B2 (0.67) CYP11B2CYP11B1PDE10A
SCHEMBL10175445 0.75 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL17896705 0.74 CYP11B2 (0.54) CYP11B2CYP11B1DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed