SCHEMBL17899652

SCHEMBL17899652

CN1CCN(c2ccc(-c3ccc(S(=O)(=O)N4CC=C(C(=O)NOC5CCCCO5)C4)cc3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 2/20 0.38
LMNA P02545 2/20 0.36
THRB P10828 1/20 0.36
RAD52 P43351 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPK1 P28482 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
TSHR P16473 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
BLM P54132 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17899695 0.93 ALDH1A1 (0.43) ALDH1A1MEN1PKMKMT2ASMN1; SMN2
SCHEMBL17897343 0.92 USP9X (0.39) ALDH1A1MEN1PKMKMT2ASMN1; SMN2
SCHEMBL17899665 0.86 KMT2A (0.44) ALDH1A1MEN1KMT2AGAALMNA
SCHEMBL17899692 0.86 PKM (0.46) ALDH1A1MEN1PKMKMT2ASMN1; SMN2
SCHEMBL17899699 0.86 KMT2A (0.39) MEN1PKMKMT2ASMN1; SMN2GAA
SCHEMBL17899697 0.85 LMNA (0.43) ALDH1A1MEN1PKMKMT2AGAA
SCHEMBL17899651 0.83 SMYD3 (0.40) ALDH1A1PKMSMN1; SMN2GAALMNA
SCHEMBL17899694 0.83 PKM (0.48) ALDH1A1MEN1PKMKMT2ASMN1; SMN2
SCHEMBL17899650 0.83 KMT2A (0.46) ALDH1A1MEN1KMT2AGAALMNA
SCHEMBL17899649 0.83 KMT2A (0.41) MEN1PKMKMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016107544-A1 INTERMEDIATE COMPOUND FOR PREPARING PYRROLE AMIDE COMPOUND AND PREPARATION METHOD AND USE THEREOF 成都先导药物开发有限公司 2016-07-07 WO disclosed