SCHEMBL17899689

SCHEMBL17899689

COc1cccc(S(=O)(=O)N2CC=C(C(=O)NOC3CCCCO3)C2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.41
PKM P14618 2/20 0.41
PKLR P30613 1/20 0.41
ALDH1A1 P00352 3/20 0.40
AKR1C3 P42330 2/20 0.40
HPGD P15428 2/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
GAA P10253 2/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
CHRM5 P08912 1/20 0.39
HTR6 P50406 1/20 0.39
HSD17B10 Q99714 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17899686 0.89 EPHX2 (0.44) HDAC1ALDH1A1KMT2AGAAMEN1
SCHEMBL17899694 0.89 PKM (0.48) PKMALDH1A1KMT2AGAAMEN1
SCHEMBL17899688 0.87 ALDH1A1 (0.46) PKMPKLRALDH1A1KMT2AGAA
SCHEMBL17899639 0.87 PKM (0.43) PKMALDH1A1KMT2AGAAHTR6
SCHEMBL17899690 0.86 ALDH1A1 (0.46) HDAC1PKMALDH1A1KMT2AMAPT
SCHEMBL17899692 0.86 PKM (0.46) PKMALDH1A1HPGDKMT2AGAA
SCHEMBL17899641 0.84 SMN1; SMN2 (0.45) ALDH1A1HPGDKMT2ANPC1GAA
SCHEMBL17899697 0.83 LMNA (0.43) PKMALDH1A1HPGDKMT2ANPC1
SCHEMBL17899644 0.82 MAPT (0.48) PKMPKLRALDH1A1KMT2ANPC1
SCHEMBL17899650 0.81 KMT2A (0.46) ALDH1A1KMT2AGAAMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016107544-A1 INTERMEDIATE COMPOUND FOR PREPARING PYRROLE AMIDE COMPOUND AND PREPARATION METHOD AND USE THEREOF 成都先导药物开发有限公司 2016-07-07 WO disclosed