SCHEMBL17899690

SCHEMBL17899690

COc1ccc(S(=O)(=O)N2CC=C(C(=O)NOC3CCCCO3)C2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
EPHX2 P34913 1/20 0.46
TSHR P16473 1/20 0.44
LMNA P02545 1/20 0.44
PKM P14618 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.43
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17899694 0.88 PKM (0.48) ALDH1A1EPHX2TSHRPKMSMN1; SMN2
SCHEMBL17899689 0.86 HDAC1 (0.41) ALDH1A1LMNAPKMHDAC1MAPT
SCHEMBL17899697 0.86 LMNA (0.43) ALDH1A1EPHX2LMNAPKMMAPT
SCHEMBL17899692 0.85 PKM (0.46) ALDH1A1EPHX2LMNAPKMSMN1; SMN2
SCHEMBL17899644 0.84 MAPT (0.48) ALDH1A1EPHX2TSHRLMNAPKM
SCHEMBL17899686 0.84 EPHX2 (0.44) ALDH1A1EPHX2HDAC1KMT2A
SCHEMBL17899650 0.84 KMT2A (0.46) ALDH1A1EPHX2LMNAMAPTKMT2A
SCHEMBL17899642 0.84 MAPT (0.39) ALDH1A1EPHX2LMNAPKMMAPT
SCHEMBL17899649 0.84 KMT2A (0.41) EPHX2PKMMAPTSMN1; SMN2KMT2A
SCHEMBL17897332 0.84 EPHX2 (0.41) ALDH1A1EPHX2SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016107544-A1 INTERMEDIATE COMPOUND FOR PREPARING PYRROLE AMIDE COMPOUND AND PREPARATION METHOD AND USE THEREOF 成都先导药物开发有限公司 2016-07-07 WO disclosed