SCHEMBL17902016

SCHEMBL17902016

O=C1N2CCCC[C@H]2CNC12CCC2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
HSD11B1 P28845 10/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 1/20 0.34
BRCA1 P38398 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GAA P10253 1/20 0.32
HTR6 P50406 1/20 0.31
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17901983 0.95 ALDH1A1 (0.35) ALDH1A1HSD11B1MEN1KMT2AMAPT
SCHEMBL23227409 0.71 MEN1 (0.37) ALDH1A1HSD11B1MEN1KMT2AMAPT
SCHEMBL2301177 0.70 HSD11B1 (0.51) HSD11B1
SCHEMBL24603324 0.70 MEN1 (0.44) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL2521564 0.70 MEN1 (0.44) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL3080507 0.66 HTR6 (0.41) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL3087078 0.66 HTR6 (0.41) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL27163373 0.66 GAA (0.41) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL18689264 0.66 HTR6 (0.41) ALDH1A1MEN1KMT2AMAPTBRCA1
SCHEMBL31207652 0.64 MEN1 (0.45) ALDH1A1HSD11B1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106629-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed