SCHEMBL23227409

SCHEMBL23227409

C[C@]1(CO)NC[C@@H]2CCCCN2C1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
BRCA1 P38398 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TYMP P19971 2/20 0.35
ALDH1A1 P00352 2/20 0.34
HSD11B1 P28845 7/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.31
CDA P32320 1/20 0.31
GAA P10253 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17901983 0.72 ALDH1A1 (0.35) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL17902016 0.71 ALDH1A1 (0.34) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL31207652 0.68 MEN1 (0.45) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL24603324 0.65 MEN1 (0.44) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL2521564 0.65 MEN1 (0.44) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL3069788 0.65 ALDH1A1 (0.40) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL1069501 0.64 HSD11B1 (0.40) MEN1KMT2AL3MBTL1TYMPALDH1A1
SCHEMBL360466 0.62 HSD11B1 (0.49) ALDH1A1HSD11B1LMNAGAA
SCHEMBL3080507 0.61 HTR6 (0.41) MEN1MAPTKMT2ABRCA1ATM
SCHEMBL3087078 0.61 HTR6 (0.41) MEN1MAPTKMT2ABRCA1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021071832-A1 ARYL HETEROBICYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. SHAW RESEARCH, LLC (US) 2021-04-15 WO disclosed