SCHEMBL17907965

SCHEMBL17907965

O=C1CCc2cc3ccc(Cl)cc3n2C1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.48
HTR2C P28335 2/20 0.48
NOTUM Q6P988 2/20 0.39
KMT2A Q03164 1/20 0.35
TDP2 O95551 3/20 0.34
KMO O15229 2/20 0.34
MAT2A P31153 2/20 0.33
DAO P14920 1/20 0.32
CTSG P08311 1/20 0.31
CMA1 P23946 1/20 0.31
F11 P03951 1/20 0.31
AHR P35869 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907930 0.87 HTR2A (0.48) HTR2AHTR2CNOTUMKMT2AF11
SCHEMBL235219 0.78 NOTUM (0.59) HTR2AHTR2CNOTUM
SCHEMBL17907947 0.77 ALDH1A1 (0.38) NOTUMKMT2ATDP2MAT2A
SCHEMBL9735956 0.77 NOTUM (0.62) HTR2AHTR2CNOTUMKMT2ATDP2
SCHEMBL17907932 0.71 SIGMAR1 (0.41) HTR2AHTR2CNOTUMRXFP1
SCHEMBL17907920 0.68 HTR2A (0.51) HTR2AHTR2CKMT2A
SCHEMBL19921327 0.66 HTR2A (0.56) HTR2AHTR2CKMT2AMAT2A
SCHEMBL17907979 0.65 PTGDR2 (0.39) HTR2AHTR2CNOTUMKMT2AKMO
SCHEMBL5619809 0.65 HTR2C (1.00) HTR2AHTR2C
SCHEMBL1770250 0.64 NOTUM (0.35) NOTUMDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed