SCHEMBL17970193

SCHEMBL17970193

Cc1cc2c(s1)C(O)CCC2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UGT2B17 O75795 2/20 0.40
PNMT P11086 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
TSHR P16473 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
PGR P06401 1/20 0.31
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13303500 0.95 UGT2B17 (0.35) UGT2B17PNMTALDH1A1HPGDTSHR
SCHEMBL13303507 0.77 UGT2B17 (0.33) UGT2B17
SCHEMBL11987736 0.77 UGT2B17 (0.33) UGT2B17ALDH1A1SMN1; SMN2
SCHEMBL11987801 0.77 HPGD (0.35) UGT2B17ALDH1A1HPGDTSHRSMN1; SMN2
SCHEMBL19981500 0.73 ADRA2A (0.31)
SCHEMBL19981792 0.73 ALDH1A1 (0.33) PNMTALDH1A1HPGDTSHRSMN1; SMN2
SCHEMBL12894433 0.73 CNR2 (0.31) UGT2B17
SCHEMBL11987727 0.73 ALDH1A1 (0.32) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL11987814 0.73 NPC1 (0.38) ALDH1A1HPGDTSHRSMN1; SMN2NPC1
SCHEMBL2837067 0.73 QDPR (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2365970-B1 PYRIDAZINONES AND THEIR USE AS BTK INHIBITORS GILEAD CONNECTICUT INC (US) 2018-03-21 EP disclosed
EP-2188267-B1 SUBSTITUTED AMIDES, METHODS OF MAKING, USE THEREOF FOR THE TREATMENT OF DISEASES SUCH AS CANCER GILEAD CONNECTICUT INC (US) 2016-08-03 EP disclosed