SCHEMBL17993486

SCHEMBL17993486

Nc1ccccc1N1C(=O)c2ccccc2N(c2ccccc2N=O)C(=O)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPA1A P0DMV8 1/20 0.41
PABPC1 P11940 1/20 0.41
SCN2A Q99250 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 3/20 0.39
GAA P10253 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 3/20 0.37
CES2 O00748 1/20 0.37
BCHE P06276 1/20 0.37
CES1 P23141 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
POLB P06746 1/20 0.36
DPP4 P27487 1/20 0.36
CYP3A4 P08684 1/20 0.36
NFKB1 P19838 1/20 0.36
PMP22 Q01453 1/20 0.36
ADORA2A P29274 1/20 0.35
MAPT P10636 2/20 0.34
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19380493 0.92 HSPA1A (0.35) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL18475716 0.86 KMT2A (0.44) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL29395615 0.77 SCN2A (0.57) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL885606 0.77 SCN2A (0.57) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL17993531 0.77 LMNA (0.50) SCN2AKMT2AMEN1KDM4EALDH1A1
SCHEMBL18470136 0.71 KMT2A (0.47) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL17993493 0.70 SCN2A (0.50) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL17993459 0.70 SCN2A (0.43) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL21942500 0.69 GAA (0.48) HSPA1APABPC1SCN2AKMT2AMEN1
SCHEMBL28247030 0.69 TLR9 (0.64) ALDH1A1NPSR1HTTTDP1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054498-A1 Bisimidazodiazocines Idemitsu Kosan Co., Ltd. (JP) 2016-08-10 EP disclosed