SCHEMBL18015353

SCHEMBL18015353

C1=CC(c2cc(-c3ccccc3-c3ccc(-c4ccccc4)nc3)cc(-c3ccccc3-c3ccc(-c4ccccn4)nc3)c2)=C(c2ccc(-c3ccccc3)nc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 4/20 0.39
P4HTM Q9NXG6 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHEK2 O96017 1/20 0.33
KDR P35968 1/20 0.33
TGFBR1 P36897 2/20 0.33
DHODH Q02127 1/20 0.33
PDK2 Q15119 1/20 0.33
CYP2A6 P11509 1/20 0.33
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CNR2 P34972 1/20 0.32
LDHA P00338 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
HSD17B1 P14061 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18573199 0.88 CHRNB2 (0.34) HPGDSCHRNB2CHRNA3LDHAHSD17B1
SCHEMBL19794441 0.82 HPGDS (0.52) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL18015360 0.79 HPGDS (0.49) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL21125929 0.78 CHEK2 (0.49) HPGDSP4HTMCHRNB2CHRNA3CHEK2
SCHEMBL20068613 0.78 CHEK2 (0.48) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL21125828 0.77 CHEK2 (0.49) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL12925598 0.77 KDM4E (0.52) HPGDSP4HTMCHEK2TGFBR1PDK2
SCHEMBL21397867 0.76 HPGDS (0.47) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL21125087 0.76 HSD17B1 (0.49) HPGDSP4HTMCHEK2KDRTGFBR1
SCHEMBL21721920 0.75 LDHA (0.50) HPGDSDHODHLDHACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016124304-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-08-11 WO disclosed