SCHEMBL18040239

SCHEMBL18040239

O=C(O)c1cn(C2CC2)c(Br)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.37
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
KDM4E B2RXH2 4/20 0.32
ALOX15 P16050 2/20 0.32
TSHR P16473 2/20 0.32
ACMSD Q8TDX5 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
WDR5 P61964 1/20 0.32
MAP3K14 Q99558 1/20 0.32
TOP2A P11388 2/20 0.32
TOP2B Q02880 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP11B2 P19099 1/20 0.32
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
GAA P10253 1/20 0.31
EPHX2 P34913 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18040241 0.93 RXFP1 (0.36) RXFP1PTGS1PTGS2KDM4EALOX15
SCHEMBL1268994 0.75 WDR5 (0.36) RXFP1PTGS1PTGS2KDM4EHCAR2
SCHEMBL25274273 0.71 RXFP1 (0.42) RXFP1PTGS1PTGS2KDM4EALOX15
SCHEMBL375420 0.69 RXFP1 (0.45) RXFP1PTGS1PTGS2KDM4EALOX15
SCHEMBL34469503 0.66 HSD17B10 (0.38) KDM4EHCAR2TOP2ATOP2BALDH1A1
SCHEMBL28041713 0.66 RXFP1 (0.41) RXFP1PTGS1PTGS2KDM4EALOX15
SCHEMBL28041712 0.66 RXFP1 (0.41) RXFP1PTGS1PTGS2KDM4EALOX15
SCHEMBL4803883 0.65 HCAR2 (0.36) KDM4EHCAR2ALDH1A1HSD17B10GAA
SCHEMBL25374471 0.64 HSD17B10 (0.40) ALDH1A1CYP11B2HSD17B10GAANOTUM
SCHEMBL70303 0.63 SMYD3 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3064502-A1 IMIDAZOPYRROLIDINONE COMPOUNDS Novartis AG (CH) 2016-09-07 EP disclosed