SCHEMBL18049433

SCHEMBL18049433

Cc1cc(C2=C(c3ccccc3)C(=O)NC2=O)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.57
GSK3B P49841 9/20 0.47
DAPK3 O43293 1/20 0.47
NTRK1 P04629 1/20 0.47
PIM1 P11309 1/20 0.47
FLT3 P36888 1/20 0.47
ROCK1 Q13464 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
POLB P06746 1/20 0.40
CASP6 P55212 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18049419 0.86 PTGS2 (0.60) PTGS2GSK3B
SCHEMBL3815134 0.78 PTGS2 (0.65) PTGS2GSK3BPOLB
SCHEMBL5762155 0.78 ACHE (0.48) PTGS2GSK3BDAPK3NTRK1PIM1
SCHEMBL114611 0.78 PTGS2 (0.67) PTGS2GSK3B
SCHEMBL3822129 0.77 PTGS2 (0.57) PTGS2GSK3B
SCHEMBL18049424 0.77 PTGS2 (0.57) PTGS2GSK3BCLK4
SCHEMBL9474080 0.75 PTGS2 (0.64) PTGS2GSK3B
SCHEMBL3816794 0.74 GSK3B (0.67) PTGS2GSK3B
SCHEMBL9237602 0.74 PTGS2 (0.54) PTGS2GSK3B
SCHEMBL934146 0.74 GSK3B (0.65) PTGS2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016144352-A2 THERAPEUTIC COMPOSITIONS INCLUDING ACRYLAMIDO COMPOUNDS OR PHENYL-SUBSTITUTED MALEIMIDE COMPOUNDS, VARIANTS THEREOF AND METHODS OF USING THE SAME STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2016-09-15 WO disclosed