SCHEMBL18052197

SCHEMBL18052197

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nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 3/20 0.54
CYP1A2 P05177 1/20 0.42
ENPEP Q07075 2/20 0.41
GLRA1 P23415 1/20 0.38
SLC6A9 P48067 1/20 0.38
OR51E2 Q9H255 1/20 0.38
LTA4H P09960 1/20 0.38
SLC7A5 Q01650 1/20 0.37
CACNA2D1 P54289 2/20 0.37
FOLH1 Q04609 2/20 0.37
NAALAD2 Q9Y3Q0 2/20 0.37
CACNB3 P54284 1/20 0.37
CACNA1C Q13936 1/20 0.37
PGR P06401 1/20 0.37
ADRA1A P35348 1/20 0.37
HTR2B P41595 1/20 0.37
CACNA2D2 Q9NY47 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1177351 1.00 GABRR1 (0.54) GABRR1CYP1A2ENPEPGLRA1SLC6A9
Hydrochloric Acid SCHEMBL28487836 0.97 GABRR1 (0.52) GABRR1CYP1A2ENPEPGLRA1SLC6A9
Trichloroacetic Acid SCHEMBL22607625 0.87 GABRR1 (0.43) GABRR1CYP1A2ENPEPLTA4HCACNA2D1
SCHEMBL9328436 0.86 GABRR1 (0.48) GABRR1CYP1A2ENPEPFOLH1NAALAD2
Methyl Aminolevulinate SCHEMBL31080862 0.81 LMNA (0.67) GABRR1CYP1A2
SCHEMBL27571000 0.80 KDM4E (0.44) GABRR1CYP1A2ENPEPFOLH1NAALAD2
SCHEMBL6905507 0.79 CYP2C19 (0.46) GABRR1CYP1A2SLC7A5FOLH1NAALAD2
SCHEMBL9736766 0.79 TDP1 (0.45) GABRR1CYP1A2ENPEPFOLH1NAALAD2
SCHEMBL6889464 0.78
SCHEMBL27867988 0.78 GABRR1 (0.43) GABRR1ENPEPGLRA1SLC6A9OR51E2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9822080-B2 Nα, Nα, Nα-trialkyl histidine derivatives useful for the preparation of ergothioneine compounds MIRONOVA INNOVATIONS, LLC (US) 2017-11-21 US disclosed
US-20170050933-A1 Nalpha, Nalpha, Nalpha-TRIALKYL HISTIDINE DERIVATIVES USEFUL FOR THE PREPARATION OF ERGOTHIONEINE COMPOUNDS Trampota Jan (US) 2017-02-23 US disclosed
US-20160264530-A1 NALPHA, NALPHA, NALPHA-TRIALKYL HISTIDINE DERIVATIVES USEFUL FOR THE PREPARATION OF ERGOTHIONEINE COMPOUNDS MIRONOVA INNOVATIONS, LLC 2016-09-15 US disclosed
US-9428463-B1 Nα, Nα, Nα-trialkyl histidine derivatives useful for the preparation of ergothioneine compounds MIRONOVA INNOVATIONS, LLC (US) 2016-08-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170050933-A1 Nalpha, Nalpha, Nalpha-TRIALKYL HISTIDINE DERIVATIVES USEFUL FOR THE PREPARATION OF ERGOTHIONEINE COMPOUNDS HNMT, TTPA, FTH1 GABRR1 2964/4885CYP1A2 1742/4885ENPEP 52/4885
US-20160264530-A1 NALPHA, NALPHA, NALPHA-TRIALKYL HISTIDINE DERIVATIVES USEFUL FOR THE PREPARATION OF ERGOTHIONEINE COMPOUNDS HNMT, TTPA, FTH1 GABRR1 2964/4885CYP1A2 1742/4885ENPEP 52/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.