SCHEMBL1817861

SCHEMBL1817861

CCS(=O)(=O)Cc1cc(NC(C)=O)ccc1S(=O)(=O)Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
CDK1 P06493 1/20 0.45
HPGD P15428 1/20 0.44
RORC P51449 1/20 0.42
ATAD2 Q6PL18 1/20 0.41
CECR2 Q9BXF3 1/20 0.41
POLB P06746 4/20 0.40
RAB9A P51151 2/20 0.40
NR4A1 P22736 1/20 0.40
ENPP2 Q13822 1/20 0.40
NPC1 O15118 2/20 0.40
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAOA P21397 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1817574 0.88 ALDH1A1 (0.53) ALDH1A1CDK1HPGDRORCATAD2
SCHEMBL1819456 0.76 CYP2C9 (0.40) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL539699 0.76 ALDH1A1 (0.73) ALDH1A1CDK1ATAD2CECR2RAB9A
SCHEMBL686781 0.75 ALDH1A1 (0.54) ALDH1A1CDK1ATAD2CECR2RAB9A
SCHEMBL6770516 0.75 ALDH1A1 (0.54) ALDH1A1CDK1ATAD2CECR2RAB9A
SCHEMBL6771522 0.73 ALDH1A1 (0.59) ALDH1A1CDK1ATAD2CECR2POLB
SCHEMBL10719928 0.73 ATAD2 (0.65) ALDH1A1CDK1RORCATAD2CECR2
SCHEMBL2436014 0.72 RORC (0.66) ALDH1A1CDK1RORCPOLBMAPT
SCHEMBL1816870 0.72 CYP1A2 (0.44) MAPTSMN1; SMN2CA12CA1CA2
SCHEMBL2535835 0.71 ALDH1A1 (0.50) ALDH1A1CDK1HPGDPOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461134-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2013-06-11 US disclosed
US-20110172187-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-07-14 US disclosed
WO-2011060196-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-05-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110172187-A1 BORON-CONTAINING SMALL MOLECULES BCL6B, BCL6, BTD ALDH1A1 4190/4885CDK1 2617/4885HPGD 4100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.