SCHEMBL1819205

SCHEMBL1819205

COC(=O)c1cc(NC(=O)C(F)(F)F)cnc1S(=O)(=O)Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CDK1 P06493 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
RORC P51449 1/20 0.36
ABL1 P00519 1/20 0.36
SRC P12931 1/20 0.36
ATF1 P18846 1/20 0.36
NFKB1 P19838 1/20 0.36
PDK1 Q15118 2/20 0.35
PDK2 Q15119 2/20 0.35
PDK3 Q15120 2/20 0.35
PDK4 Q16654 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1818375 0.85 RORC (0.40) CYP1A2CYP2C9CYP2C19L3MBTL1CA12
SCHEMBL1818471 0.80 AR (0.41) L3MBTL1CA12CA1CA2CA9
SCHEMBL8325235 0.80 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19L3MBTL1IDO1
SCHEMBL1816743 0.77 ABCC9 (0.40) CYP2C19CA12CA1CA2CA9
SCHEMBL19682925 0.75 OPRK1 (0.44) L3MBTL1ABL1KDM4E
SCHEMBL19682732 0.74 OPRK1 (0.46)
SCHEMBL1819819 0.72 CA1 (0.45) CA12CA1CA2CA9
SCHEMBL8321765 0.70 PDK1 (0.45) CYP1A2CYP2C9CYP2C19ATF1NFKB1
SCHEMBL1819520 0.70 PKM (0.57) CYP1A2CYP2C9CYP2C19L3MBTL1ABL1
SCHEMBL18247535 0.70 ATM (0.53) CYP1A2CYP2C9CYP2C19L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212918-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-09-01 US disclosed
WO-2011060199-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-05-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212918-A1 BORON-CONTAINING SMALL MOLECULES BCL6B, BCL6, BTD CYP1A2 3504/4885CYP2C9 3001/4885CYP2C19 3226/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.