SCHEMBL18212

SCHEMBL18212

Cn1c(-c2nccc(C(F)(F)F)n2)noc1=O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.37
IDH1 O75874 6/20 0.36
IDH2 P48735 4/20 0.36
MBOAT4 Q96T53 1/20 0.36
KCNT1 Q5JUK3 4/20 0.35
ADRB1 P08588 1/20 0.34
HDAC4 P56524 2/20 0.33
KCNQ1 P51787 1/20 0.33
KCNH2 Q12809 1/20 0.33
CACNA1C Q13936 1/20 0.33
SCN5A Q14524 1/20 0.33
KCNMB1 Q16558 1/20 0.33
KCNT2 Q6UVM3 1/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 1/20 0.33
HSP90AA1 P07900 1/20 0.33
RAB9A P51151 1/20 0.33
S1PR1 P21453 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18577 0.76 IDH1 (0.39) IDH1IDH2KCNT1KDM4ENPC1
SCHEMBL2334760 0.73 NPSR1 (0.42) P2RX7ADRB1KDM4ENPC1RAB9A
SCHEMBL18484 0.71 CA2 (0.38) KCNT1KDM4EPTGS2
SCHEMBL18781 0.69 ALDH1A1 (0.38) IDH1IDH2ADRB1HDAC4
SCHEMBL22271284 0.67 IDH1 (0.50) P2RX7IDH1IDH2MBOAT4ADRB1
SCHEMBL16986457 0.66 IDH1 (0.38) P2RX7IDH1IDH2KCNT1ADRB1
SCHEMBL9771829 0.65 NPC1 (0.44) KDM4ENPC1RAB9A
SCHEMBL22637946 0.65 IDH1 (0.45) IDH1IDH2KCNT1KCNQ1KCNH2
SCHEMBL22637944 0.65 IDH1 (0.45) IDH1IDH2KCNT1KCNQ1KCNH2
SCHEMBL22637369 0.64 KCNT1 (0.53) KCNT1KCNQ1KCNH2CACNA1CSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025460-A1 OXADIAZOLINONE DERIVATIVES AND USE THEREOF IN PEST CONTROL BAYER CROPSCIENCE AG (DE) 2012-03-01 WO disclosed