SCHEMBL18214697

SCHEMBL18214697

CCCC(=N)n1c(=N)c(=O)[nH]c2cc(C(=O)N3CCN(C)C(c4ccccc4)C3)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.42
HSD17B10 Q99714 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
THRB P10828 1/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
MGLL Q99685 1/20 0.38
RAB9A P51151 3/20 0.37
HSP90AA1 P07900 3/20 0.37
NPC1 O15118 1/20 0.37
PARP1 P09874 1/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 3/20 0.37
PKM P14618 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
AURKB Q96GD4 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1726455 0.76 GRIN2D (0.46) P2RX7HSD17B10MEN1POLBTHRB
SCHEMBL18214696 0.74 SMN1; SMN2 (0.42) HSD17B10MEN1POLBTHRBTSHR
SCHEMBL18214723 0.73 BRPF1 (0.43) MEN1THRBKMT2AALDH1A1KDM4E
SCHEMBL18214707 0.72 TP53 (0.46) HSD17B10MEN1KMT2AHSP90AA1PARP1
SCHEMBL7907649 0.70 ALDH1A1 (0.44) P2RX7HSD17B10MEN1POLBTHRB
SCHEMBL10186595 0.69 POLB (0.41) HSD17B10MEN1POLBTHRBTSHR
SCHEMBL7905362 0.69 RAB9A (0.42) P2RX7HSD17B10MEN1POLBTHRB
SCHEMBL17706167 0.67
SCHEMBL15217072 0.66
SCHEMBL3274315 0.64 P2RX7 (0.55) P2RX7MEN1POLBTSHRRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2404922-B1 QUINOXALINE COMPOUNDS ASTELLAS PHARMA INC (JP) 2016-11-09 EP disclosed