Decoquinate

Decoquinate

SCHEMBL18227083

CCCCCCCCCCOc1cc2c(O)c(C(=O)OCC)cnc2cc1OCC.CCCc1ncc(C[n+]2ccccc2C)c(N)n1.[Cl-]

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Decoquinate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.53
KDM4E B2RXH2 1/20 0.53
SLC19A2 O60779 1/20 0.53
USP2 O75604 1/20 0.53
CASP1 P29466 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
TP53 P04637 1/20 0.34
PDPK1 O15530 1/20 0.34
DPP4 P27487 3/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
TSHR P16473 1/20 0.32
AGTR1 P30556 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Decoquinate SCHEMBL29373625 0.77 DPP4 (0.46) LMNAKDM4ENPC1RAB9AHSD17B10
Decoquinate SCHEMBL43853 0.77 DPP4 (0.46) LMNAKDM4ENPC1RAB9AHSD17B10
Decoquinate SCHEMBL14247781 0.75 DPP4 (0.44) LMNAKDM4ENPC1RAB9AHSD17B10
Decoquinate SCHEMBL14247780 0.75 DPP4 (0.44) LMNANPC1RAB9AHSD17B10SMN1; SMN2
Decoquinate SCHEMBL15152849 0.75 LMNA (0.47) LMNAKDM4ENPC1RAB9AHSD17B10
Amprolium Ion SCHEMBL29910331 0.73 KDM4E (0.98) LMNAKDM4ESLC19A2USP2CASP1
Amprolium Ion SCHEMBL362893 0.73 KDM4E (0.98) LMNAKDM4ESLC19A2USP2CASP1
Decoquinate SCHEMBL10696854 0.73 DPP4 (0.42) LMNAKDM4ENPC1RAB9AHSD17B10
Amprolium Ion SCHEMBL29737311 0.73 KDM4E (1.00) LMNAKDM4ESLC19A2USP2CASP1
Amprolium Ion SCHEMBL363586 0.73 KDM4E (0.95) LMNAKDM4ESLC19A2USP2CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016181187-A1 COMPOSITION FOR THE TREATMENT OF GREGARINE INFESTATION IN SHRIMP LABORATORIO AVI-MEX, S.A. DE C.V. (MX) 2016-11-17 WO disclosed