SCHEMBL1828068

SCHEMBL1828068

COc1ccc2c(c1OC)N=CCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
LMNA P02545 1/20 0.38
ACHE P22303 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 2/20 0.37
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
DRD2 P14416 3/20 0.34
PTGS2 P35354 1/20 0.34
PDE1B Q01064 6/20 0.34
PDE2A O00408 1/20 0.34
PDE8B O95263 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR2B P41595 1/20 0.34
PDE1A P54750 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE1C Q14123 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25895759 0.77 HTR5A (0.41) DRD2PTGS2DRD1
SCHEMBL31061252 0.77 HTR5A (0.41) DRD2PTGS2DRD1
SCHEMBL9404873 0.75 KDM4E (0.40) KDM4ELMNAACHEALDH1A1HPGD
SCHEMBL9404804 0.72 NPC1 (0.43) KDM4ELMNAACHEALDH1A1HPGD
SCHEMBL30203107 0.68 MAOB (0.35) KDM4EALDH1A1MAPTCYP3A4
SCHEMBL3158365 0.66 KDM4E (0.56) KDM4ELMNAACHEALDH1A1HPGD
SCHEMBL1828066 0.66 MAPT (0.45) KDM4ELMNAALDH1A1MAPTKMT2A
SCHEMBL28227231 0.65 DRD2 (0.36) KDM4EHPGDDRD2DRD1
SCHEMBL3674074 0.65 CA9 (0.50) KDM4EACHEALDH1A1HPGDMAPT
SCHEMBL30701949 0.65 CA9 (0.50) KDM4EACHEALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315614-A1 CATIONIC DIHYDROISOQUINOLINIUM DERIVATIVES FOR USE AS BLEACH ACTIVATORS Henkel AG & Co. KGaA (DE) 2011-05-04 EP disclosed
WO-2010022995-A1 CATIONIC DIHYDROISOQUINOLINIUM DERIVATIVES FOR USE AS BLEACH ACTIVATORS HENKEL AG & CO. KGAA (DE) 2010-03-04 WO disclosed