SCHEMBL18285697

SCHEMBL18285697

CC(C)N(CCC(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 3/20 0.37
CA1 P00915 3/20 0.37
CA12 O43570 2/20 0.37
CA7 P43166 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
CA2 P00918 2/20 0.35
NAALAD2 Q9Y3Q0 1/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
EPHX2 P34913 1/20 0.34
KDM4C Q9H3R0 2/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
KDM4A O75164 1/20 0.33
PHF8 Q9UPP1 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18281954 0.86 CTSS (0.34) CA14CA1CA12CA7HDAC6
SCHEMBL23564375 0.85 CTSL (0.37) CA14CA1CA7HDAC6HDAC1
SCHEMBL29023150 0.85 CA14 (0.35) CA14CA1CA12CA7HDAC6
SCHEMBL20721672 0.84 HDAC6 (0.36) CA14CA1CA12CA7HDAC6
SCHEMBL5724032 0.83 HDAC6 (0.34) CA14CA1CA12CA7HDAC6
SCHEMBL21175428 0.81 CTSS (0.39) CA14HDAC6HDAC1HDAC2CTSS
SCHEMBL21175429 0.81 CTSS (0.39) CA14HDAC6HDAC1HDAC2CTSS
SCHEMBL1067066 0.81 CA14 (0.38) CA14CA1CA12CA7HDAC6
SCHEMBL3469119 0.81 CA14 (0.46) CA14CA1CA12CA7HDAC6
SCHEMBL18202365 0.80 CA14 (0.39) CA14CA1CA12CA7HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025049064-A9 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC. (US) 2025-05-22 WO disclosed
WO-2025049064-A2 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC. (US) 2025-03-06 WO disclosed
US-20240270765-A2 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC. 2024-08-15 US disclosed
US-20240025928-A1 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC (US) 2024-01-25 US disclosed
US-20240025928-A1 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC (US) 2024-01-25 US disclosed
US-20240025928-A1 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE SIGNPATH PHARMA INC (US) 2024-01-25 US disclosed
US-11661403-B2 Oxadiazole compounds VIVACE THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-11661403-B2 Oxadiazole compounds VIVACE THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-11661403-B2 Oxadiazole compounds VIVACE THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-20230144106-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY SYROS PHARMACEUTICALS INC (US) 2023-05-11 US disclosed
US-20210221820-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY SYROS PHARMACEUTICALS INC (US) 2021-07-22 US disclosed
US-20210188833-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY SYROS PHARMACEUTICALS INC (US) 2021-06-24 US disclosed
EP-3793551-A1 OXADIAZOLE COMPOUNDS Vivace Therapeutics, Inc. (US) 2021-03-24 EP disclosed
WO-2019222431-A9 OXADIAZOLE COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2020-10-22 WO disclosed
WO-2019222431-A9 OXADIAZOLE COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2020-10-22 WO disclosed
US-10787444-B2 Compounds for the modulation of myc activity SYROS PHARMACEUTICALS, INC. (US) 2020-09-29 US disclosed
US-20190048019-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY OXFORD FINANCE LLC, AS COLLATERAL AGENT 2019-02-14 US disclosed
US-20180162851-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY OXFORD FINANCE LLC, AS COLLATERAL AGENT 2018-06-14 US disclosed
US-20180162851-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY OXFORD FINANCE LLC, AS COLLATERAL AGENT 2018-06-14 US disclosed
WO-2016197078-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY SYROS PHARMACEUTICALS, INC. (US) 2016-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180162851-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY MYC, MYCBP, MYCBP2 CA14 1628/4885CA1 2709/4885CA12 1740/4885
US-20190048019-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY MYC, MYCBP, MYCBP2 CA14 1546/4885CA1 2980/4885CA12 1772/4885
US-20240025928-A1 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE CPT1B, FABP3, NR1H2 CA14 3229/4885CA1 1338/4885CA12 2143/4885
US-20240270765-A2 CARDIOPROTECTIVE LIPIDS AND METHODS OF USE CPT1B, FABP3, NR1H2 CA14 3229/4885CA1 1338/4885CA12 2143/4885
US-20210188833-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY MYC, MYCBP, MYCBP2 CA14 1449/4885CA1 3057/4885CA12 1629/4885
US-20230144106-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY MYC, MYCBP, MYCBP2 CA14 1449/4885CA1 3057/4885CA12 1629/4885
US-10787444-B2 Compounds for the modulation of myc activity MYC, MYCBP, MYCBP2 CA14 1628/4885CA1 2709/4885CA12 1740/4885
US-20210221820-A1 COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY MYC, MYCBP, MYCBP2 CA14 1546/4885CA1 2980/4885CA12 1772/4885
US-11661403-B2 Oxadiazole compounds YAP1, TEAD2, TEAD3 CA14 4632/4885CA1 4666/4885CA12 4453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.