SCHEMBL1832039

SCHEMBL1832039

O=C(O)c1ccc(F)cc1N1C(=O)CC(O)C1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 6/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 9/20 0.38
KEAP1 Q14145 1/20 0.37
MAPT P10636 7/20 0.36
HTR7 P34969 1/20 0.36
GAA P10253 4/20 0.35
LMNA P02545 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
NLRP1 Q9C000 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
P2RX7 Q99572 1/20 0.33
HSD17B10 Q99714 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1834304 0.83 PKM (0.36) PKMKDM4EALDH1A1MAPTGAA
SCHEMBL317703 0.79 KEAP1 (0.43) KDM4EALDH1A1KEAP1HTR7GAA
SCHEMBL31653832 0.79 KEAP1 (0.43) KDM4EALDH1A1KEAP1HTR7GAA
SCHEMBL29549481 0.71 SCN2A (0.54) KDM4EALDH1A1KEAP1GAALMNA
SCHEMBL3825337 0.70 GAA (0.50) KDM4EALDH1A1KEAP1MAPTGAA
SCHEMBL3830992 0.68 KEAP1 (0.41) KDM4EALDH1A1KEAP1MAPTGAA
SCHEMBL3824501 0.68 GAA (0.55) PKMKDM4EALDH1A1GAALMNA
SCHEMBL4432960 0.67 PTPN1 (0.38) PKMKDM4EALDH1A1MAPTGAA
SCHEMBL28946278 0.66 ALDH1A1 (0.49) KDM4EALDH1A1KEAP1MAPTGAA
SCHEMBL17119924 0.66 F2RL1 (0.46) KEAP1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318366-A2 PSMA-BINDING AGENTS AND USES THEREOF The Johns Hopkins University (US) 2011-05-11 EP disclosed
WO-2010014933-A2 PSMA-BINDING AGENTS AND USES THEREOF THE JOHNS HOPKINS UNIVERSITY (US) 2010-02-04 WO disclosed