SCHEMBL1832044

SCHEMBL1832044

O=C(O)c1ccc(F)c(O)c1N1C(=O)CCC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.43
CA1 P00915 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
AKR1C2 P52895 2/20 0.38
AKR1C1 Q04828 2/20 0.38
SELL P14151 1/20 0.35
SELP P16109 1/20 0.35
TSHR P16473 2/20 0.33
CASP1 P29466 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
TTR P02766 1/20 0.33
CA2 P00918 1/20 0.33
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
CYP1A2 P05177 1/20 0.32
GRIK1 P39086 1/20 0.32
STAT3 P40763 1/20 0.32
PIM3 Q86V86 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1834310 0.81 CA12 (0.41) CA1CA12CA9SELLSELP
SCHEMBL317655 0.79 ALB (0.49) ALBCA1CA12CA9AKR1C2
SCHEMBL20837977 0.72 CA12 (0.42) CA1CA12CA9CYP1A2KMT2A
SCHEMBL4432972 0.71 ALDH1A1 (0.40) CA1CA12CA9SELLSELP
SCHEMBL13315472 0.70 ALB (0.65) ALBCA1CA12CA9AKR1C2
SCHEMBL6828586 0.70 ALB (0.53) ALBCA1AKR1C2AKR1C1SELL
SCHEMBL31455903 0.69 ALB (0.57) ALBCA1CA12CA9AKR1C2
SCHEMBL7880433 0.69 ALB (0.57) ALBCA1CA12CA9AKR1C2
SCHEMBL31653832 0.69 KEAP1 (0.43) ALBCA1CA12CA9TSHR
SCHEMBL317703 0.69 KEAP1 (0.43) ALBCA1CA12CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318366-A2 PSMA-BINDING AGENTS AND USES THEREOF The Johns Hopkins University (US) 2011-05-11 EP disclosed
WO-2010014933-A2 PSMA-BINDING AGENTS AND USES THEREOF THE JOHNS HOPKINS UNIVERSITY (US) 2010-02-04 WO disclosed