SCHEMBL18323943

SCHEMBL18323943

CC(C)C(O)CCN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP7 Q9UHL4 1/20 0.43
TRPA1 O75762 3/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
OPRK1 P41145 4/20 0.41
OPRM1 P35372 3/20 0.41
OPRD1 P41143 3/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
NCOR2 Q9Y618 2/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4798287 0.84 CARM1 (0.53) TRPA1OPRK1ALDH1A1TSHRADRA2B
SCHEMBL16653971 0.81 OPRK1 (0.45) DPP7MEN1KMT2AOPRK1OPRM1
SCHEMBL18002191 0.81 TRPA1 (0.46) TRPA1MEN1KMT2AOPRK1ALDH1A1
SCHEMBL13995266 0.81 OPRK1 (0.53) DPP7OPRK1OPRM1OPRD1ALDH1A1
SCHEMBL21227439 0.79 HDAC3 (0.47) DPP7MEN1KMT2AOPRK1OPRM1
SCHEMBL2310169 0.77 TSHR (0.51) DPP7MEN1KMT2AOPRK1OPRM1
SCHEMBL12039805 0.77 OPRK1 (0.53) MEN1KMT2AOPRK1OPRM1OPRD1
SCHEMBL9640804 0.76 TSHR (0.54) MEN1KMT2AOPRK1OPRM1OPRD1
SCHEMBL8983567 0.76 RIPK1 (0.47) DPP7OPRK1ALDH1A1TSHRHDAC3
SCHEMBL11237204 0.76 RIPK1 (0.46) DPP7MEN1KMT2AOPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2917206-B1 HETEROARYL SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL MYERS SQUIBB CO (US) 2016-12-21 EP disclosed