SCHEMBL18358995

SCHEMBL18358995

O=C(NCCC(F)(F)F)c1ccc(-c2cocn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.44
HDAC4 P56524 10/20 0.43
HDAC6 Q9UBN7 8/20 0.43
HDAC1 Q13547 5/20 0.41
HDAC3 O15379 2/20 0.41
PPARD Q03181 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
CD274 Q9NZQ7 1/20 0.39
HPGDS O60760 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976449 0.79 HDAC4 (0.48) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL16964549 0.79 NPC1 (0.47) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL16964206 0.78 KDM4E (0.43) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL19976499 0.75 MLYCD (0.46) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL19976443 0.75 HDAC4 (0.44) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL16991011 0.74 KDM4E (0.43) MLYCDHDAC4HDAC6HDAC1HDAC3
SCHEMBL16964243 0.74 KDM4E (0.54) MLYCDKDM4EALDH1A1
SCHEMBL6513323 0.74 PLOD2 (0.54) HDAC4
SCHEMBL16964231 0.74 MLYCD (0.55) MLYCDHDAC3ALDH1A1
SCHEMBL16963678 0.73 KDM4E (0.73) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900638-B1 COMPOUNDS FOR USE IN THE TREATMENT OF MYCOBACTERIAL INFECTIONS UNIVERSITÉ DE DROIT ET DE LA SANTÉ DE LILLE 2 (FR) 2017-01-04 EP disclosed