SCHEMBL19976443

SCHEMBL19976443

O=C(NCCC(F)(F)F)c1ccc(-c2ncno2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 12/20 0.44
HDAC6 Q9UBN7 11/20 0.44
SPHK2 Q9NRA0 1/20 0.43
HDAC1 Q13547 5/20 0.43
MLYCD O95822 1/20 0.43
HDAC3 O15379 3/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
S1PR1 P21453 1/20 0.39
NCOR2 Q9Y618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16965137 0.79 LMNA (0.53) HDAC4HDAC6SPHK2HDAC1MLYCD
SCHEMBL19976499 0.77 MLYCD (0.46) HDAC4HDAC6HDAC1MLYCDHDAC3
SCHEMBL16965201 0.76 MAPK14 (0.57) HDAC6MLYCD
SCHEMBL19976449 0.75 HDAC4 (0.48) HDAC4HDAC6HDAC1MLYCDHDAC3
SCHEMBL18358995 0.75 MLYCD (0.44) HDAC4HDAC6HDAC1MLYCDHDAC3
SCHEMBL16964307 0.75 PSMB8 (0.46) HDAC4HDAC6SPHK2HDAC1MLYCD
SCHEMBL16964102 0.73 PLK1 (0.61) HDAC4HDAC6HDAC1HDAC3HDAC7
SCHEMBL16964231 0.73 MLYCD (0.55) MLYCDHDAC3
SCHEMBL16964206 0.72 KDM4E (0.43) HDAC4HDAC6HDAC1MLYCDHDAC3
SCHEMBL16964142 0.71 MLYCD (0.54) MLYCDHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920042-B2 Compounds for use in the treatment of mycobacterial infections UNIVERSITE DE DROIT ET DE LA SANTE DE LILLE 2 (FR) 2018-03-20 US disclosed