SCHEMBL1839256

SCHEMBL1839256

N#Cc1ccccc1-c1ccc(Cc2nc([N+](=O)[O-])c[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.39
BRS3 P32247 2/20 0.38
RIPK1 Q13546 1/20 0.37
PPARG P37231 2/20 0.37
TRPA1 O75762 1/20 0.37
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
PTPN5 P54829 1/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA1 Q13131 2/20 0.35
PRKAB1 Q9Y478 2/20 0.35
MME P08473 1/20 0.35
MYC P01106 1/20 0.34
WDR5 P61964 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1840296 0.80 BRS3 (0.48) BRS3
SCHEMBL6054864 0.79 RIPK1 (0.51) RIPK1GRIN1GRIN2BALDH1A1
SCHEMBL1839909 0.76 BRS3 (0.48) BRS3
SCHEMBL1838065 0.73 SOS1 (0.59) PPARGPRKAG1PRKAA1PRKAB1ALDH1A1
SCHEMBL28116298 0.71 PRKAG1 (0.43) ESR2PPARGFFAR1AKR1B1PTPN5
SCHEMBL1839656 0.70 ALDH1A1 (0.47) ESR2PPARGPRKAG1PRKAA1PRKAB1
SCHEMBL7433163 0.70 ESR2 (0.56) ESR2PTPN5ALDH1A1MAPK1
SCHEMBL1890018 0.68 ESR2 (0.45) ESR2PPARGFFAR1AKR1B1PTPN5
SCHEMBL1840030 0.68 MAPT (0.67) PPARGALDH1A1
SCHEMBL1895309 0.67 KDM4E (0.41) ESR2PPARGMYCWDR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321281-A2 ANTI INFLAMMATORY COMPOUNDS Elder Pharmaceuticals Ltd (IN) 2011-05-18 EP claimed
WO-2010029576-A2 ANTI INFLAMMATORY COMPOUNDS ELDER PHARMACEUTICALS LTD. (IN) 2010-03-18 WO claimed
EP-2321281-A2 ANTI INFLAMMATORY COMPOUNDS Elder Pharmaceuticals Ltd (IN) 2011-05-18 EP disclosed
WO-2010029576-A2 ANTI INFLAMMATORY COMPOUNDS ELDER PHARMACEUTICALS LTD. (IN) 2010-03-18 WO disclosed