SCHEMBL18397802

SCHEMBL18397802

O=C(Nc1ccccc1)c1ccccc1CBr

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.70
ALDH1A1 P00352 3/20 0.66
ADRB2 P07550 1/20 0.66
CYP3A4 P08684 2/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C19 P33261 1/20 0.59
MEN1 O00255 6/20 0.58
KMT2A Q03164 6/20 0.58
HPGD P15428 2/20 0.58
KDM4E B2RXH2 2/20 0.58
LMNA P02545 2/20 0.58
TP53 P04637 2/20 0.58
HTT P42858 1/20 0.58
HSD17B10 Q99714 1/20 0.58
TDP1 Q9NUW8 1/20 0.56
METAP2 P50579 1/20 0.54
CYP2C9 P11712 1/20 0.54
ALOX12 P18054 1/20 0.54
CHRNB2 P17787 1/20 0.54
CHRNB4 P30926 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1193435 0.84 BCAT2 (0.72) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL19259498 0.84 BCAT2 (0.72) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL27819009 0.82 BCAT2 (0.70) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL1072315 0.81 ALDH1A1 (0.73) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL8971238 0.81 ALDH1A1 (0.73) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL437231 0.80 ALDH1A1 (0.87) BCAT2ALDH1A1ADRB2CYP3A4MEN1
SCHEMBL5595491 0.79 ALDH1A1 (0.71) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL27510518 0.79 ALDH1A1 (0.67) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL1441429 0.79 BCAT2 (0.60) BCAT2ALDH1A1ADRB2CYP3A4CYP1A2
SCHEMBL11266259 0.78 ALDH1A1 (0.83) BCAT2ALDH1A1ADRB2CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3325462-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF Pharmakea, Inc. (US) 2018-05-30 EP disclosed
WO-2017015221-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2017-01-26 WO disclosed