SCHEMBL18436288

SCHEMBL18436288

CC(C)Cc1ccccc1-c1ccc(C#N)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
ADRA2C P18825 1/20 0.41
MAOB P27338 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
CYP11B2 P19099 3/20 0.39
SCN10A Q9Y5Y9 1/20 0.38
TSHR P16473 1/20 0.38
IDO1 P14902 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
SLC6A4 P31645 1/20 0.37
KIF11 P52732 1/20 0.37
STAT3 P40763 1/20 0.36
CYP2A6 P11509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10590473 0.86 CYP11B2 (0.39) KMT2AADRA2CMAOBCYP11B2TSHR
SCHEMBL8472098 0.81 CYP2A6 (0.48) ADRA2CMAOBCYP11B2TSHRIDO1
SCHEMBL4935794 0.81 ADRA2C (0.44) ADRA2CMAOBCYP11B2TSHRIDO1
SCHEMBL4630258 0.80 KMT2A (0.60) KMT2AGABRA1GABRB2CYP11B2SLC6A4
SCHEMBL6162265 0.79 MMP3 (0.45) ADRA2CMAOBCYP11B2TSHRPTGDR2
SCHEMBL8632293 0.79 KMT2A (0.46) KMT2AGABRA1GABRB2
SCHEMBL11136713 0.78 CYP11B2 (0.39) ADRA2CGABRA1GABRB2CYP11B2
SCHEMBL28848262 0.78 ADRA2C (0.49) ADRA2CMAOBCYP11B2TSHRPTGDR2
SCHEMBL13873005 0.77 KMT2A (0.44) KMT2AGABRA1GABRB2SLC6A4
SCHEMBL8492143 0.77 GABRA1 (0.52) KMT2AGABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed