SCHEMBL18436681

SCHEMBL18436681

COc1c(NCCNC(=O)Cc2ccncc2)cnc2c(-c3ccc(C#N)cc3)cccc12

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.38
MAPT P10636 2/20 0.37
NAMPT P43490 1/20 0.37
POLB P06746 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
DGAT2 Q96PD7 6/20 0.36
MAP3K11 Q16584 1/20 0.36
NTRK1 P04629 1/20 0.35
PDCD1 Q15116 2/20 0.35
CD274 Q9NZQ7 2/20 0.35
KDM4A O75164 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
CNR2 P34972 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
ABCB1 P08183 1/20 0.35
HPGD P15428 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
NPY5R Q15761 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18436930 0.88 POLB (0.39) MAPTPOLBALDH1A1PDCD1CD274
SCHEMBL18436729 0.86 CD274 (0.43) ALDH1A1PDCD1CD274KDM4AKDM5B
SCHEMBL18436545 0.82 MTNR1A (0.39) GSK3BALDH1A1PDCD1CD274KDM4A
SCHEMBL21336770 0.82 EGLN1 (0.40) MAPTPOLBPDCD1CD274
SCHEMBL21336708 0.81 HTR1A (0.36) PDCD1CD274KDM4AKDM5BSLC22A12
SCHEMBL18436862 0.81 EGLN1 (0.36) PDCD1CD274KDM4AKDM5BCNR2
SCHEMBL18436919 0.81 EGLN1 (0.36) DGAT2PDCD1CD274KDM4AKDM5B
SCHEMBL18436682 0.80 RAD52 (0.38) KDM4AKDM5BSLC22A12
SCHEMBL18436737 0.79 KDM4E (0.46) POLBALDH1A1HPGD
SCHEMBL18436859 0.79 TP53 (0.44) MAPTNAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed