SCHEMBL1845523

SCHEMBL1845523

COC(=O)C[C@@](O)(CCN(CCc1ccc(Br)cc1)C(=O)OC)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37
PLAAT4 Q9UL19 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
ALOX5 P09917 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 1/20 0.35
IDO1 P14902 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
HSP90AA1 P07900 1/20 0.34
MLYCD O95822 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1845524 1.00 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL3709010 0.88 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL3709009 0.88 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL1844871 0.80 TAAR1 (0.38) PTGDR2PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL3717915 0.77 KMT2A (0.34) KMT2AMEN1TDP1ALDH1A1
SCHEMBL958964 0.77 KMT2A (0.36) KMT2AMEN1ALOX5ALDH1A1CHRM2
SCHEMBL3709505 0.77 THRA (0.46) HDAC1HDAC6PLAAT3PLAAT5PLAAT2
SCHEMBL9955949 0.76 MEN1 (0.38) HDAC1HDAC6PLAAT3PLAAT5PLAAT2
SCHEMBL1846498 0.73 TAAR1 (0.37) HDAC1HDAC6PTGDR2KMT2AMEN1
SCHEMBL735527 0.70 SMN1; SMN2 (0.34) KMT2AMEN1ALOX5ALDH1A1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324017-A2 INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1 Boehringer Ingelheim International GmbH (DE) 2011-05-25 EP disclosed
WO-2010010157-A2 INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-28 WO disclosed