SCHEMBL9955949

SCHEMBL9955949

CC(C)(O)C[C@@](O)(CCN(CCc1ccc(Br)cc1)C(=O)O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37
PLAAT4 Q9UL19 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
RCE1 Q9Y256 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HDAC1 Q13547 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
ALOX5 P09917 1/20 0.34
GPR52 Q9Y2T5 1/20 0.34
PDPK1 O15530 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
FDPS P14324 1/20 0.33
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709009 0.89 HDAC1 (0.39) MEN1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL3709010 0.89 HDAC1 (0.39) MEN1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL9955344 0.79 HSD11B1 (0.42) HDAC6
SCHEMBL1845524 0.76 HDAC1 (0.39) MEN1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL1845523 0.76 HDAC1 (0.39) MEN1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL15674404 0.76 ALOX5 (0.36) MEN1KMT2AALOX5CHRM2CHRM3
SCHEMBL9955946 0.76 ALOX5 (0.36) MEN1KMT2AALOX5CHRM2CHRM3
SCHEMBL9954703 0.76 DRD2 (0.44) PLAAT3PLAAT5PLAAT2PLAAT4TAAR1
SCHEMBL1846498 0.73 TAAR1 (0.37) MEN1KMT2ATAAR1TDP1HDAC1
SCHEMBL9954699 0.73 NR1H2 (0.41) MEN1KMT2ANPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655349-A1 METHODS OF MAKING DIASTEREOMERIC ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2013-10-30 EP disclosed
WO-2012087720-A1 METHODS OF MAKING DIASTEREOMERIC ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 WO disclosed