SCHEMBL3709010

SCHEMBL3709010

COC(=O)N(CCc1ccc(Br)cc1)CCC(O)(CC(C)(C)O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.37
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37
PLAAT4 Q9UL19 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALOX5 P09917 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
HSP90AA1 P07900 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SLC6A2 P23975 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33
LTB4R Q15722 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
LPAR1 Q92633 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709009 1.00 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL9955949 0.89 MEN1 (0.38) HDAC1HDAC6PLAAT3PLAAT5PLAAT2
SCHEMBL1845524 0.88 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL1845523 0.88 HDAC1 (0.39) HDAC1HDAC6PTGDR2PLAAT3PLAAT5
SCHEMBL1846498 0.85 TAAR1 (0.37) HDAC1HDAC6PTGDR2MEN1KMT2A
SCHEMBL1846565 0.79 ALDH1A1 (0.34) MEN1KMT2A
SCHEMBL956652 0.78 SMN1; SMN2 (0.34) MEN1KMT2AALOX5CHRM2CHRM3
SCHEMBL9954703 0.75 DRD2 (0.44) PLAAT3PLAAT5PLAAT2PLAAT4TAAR1
SCHEMBL3709505 0.74 THRA (0.46) HDAC1HDAC6PLAAT3PLAAT5PLAAT2
SCHEMBL9955077 0.72 POLB (0.46) HDAC1HDAC6PLAAT3PLAAT5PLAAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393807-A1 CYCLIC INHIBITORS OF 11 -HYDROXYSTEROID DEHYDROGENASE 1 Boehringer Ingelheim International GmbH (DE) 2011-12-14 EP disclosed
WO-2010089303-A1 CYCLIC INHIBITORS OF 11 β-HYDROXYSTEROID DEHYDROGENASE 1 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-12 WO disclosed