SCHEMBL18458019

SCHEMBL18458019

CCC(O)N(CC1(N2CCN(Cc3ccccc3)CC2)CCOCC1)c1ncccc1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.62
OPRM1 P35372 18/20 0.62
KCNH2 Q12809 9/20 0.51
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21337558 0.84 SIGMAR1 (0.73) SIGMAR1OPRM1KCNH2HSD11B1
SCHEMBL18426796 0.84 SIGMAR1 (0.89) SIGMAR1OPRM1KCNH2
SCHEMBL18458556 0.81 SIGMAR1 (0.71) SIGMAR1OPRM1KCNH2
SCHEMBL18425567 0.77 SIGMAR1 (1.00) SIGMAR1OPRM1KCNH2HSD11B1
SCHEMBL21337397 0.75 SIGMAR1 (0.50) SIGMAR1OPRM1KCNH2
SCHEMBL18458966 0.75 HSD11B1 (0.51) SIGMAR1OPRM1KCNH2HSD11B1
SCHEMBL20621716 0.74 SIGMAR1 (0.48) SIGMAR1OPRM1KCNH2
SCHEMBL18458027 0.74 SIGMAR1 (0.79) SIGMAR1OPRM1KCNH2
SCHEMBL18458533 0.74 SIGMAR1 (0.88) SIGMAR1OPRM1KCNH2
SCHEMBL18458023 0.73 OPRM1 (0.68) SIGMAR1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017016669-A1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-02-02 WO disclosed