SCHEMBL184604

SCHEMBL184604

COC(=O)Cc1ccc(S(=O)(=O)N2CCCCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.64
GLA P06280 1/20 0.63
ALDH1A1 P00352 6/20 0.63
TSHR P16473 1/20 0.63
HSD17B10 Q99714 1/20 0.63
TDP1 Q9NUW8 1/20 0.62
KMT2A Q03164 4/20 0.58
MAPT P10636 2/20 0.58
MEN1 O00255 2/20 0.58
HTT P42858 1/20 0.57
USP2 O75604 2/20 0.57
PKM P14618 1/20 0.56
LMNA P02545 1/20 0.56
POLB P06746 1/20 0.55
ATM Q13315 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623009 0.99 AGTR1 (0.62) AGTR1GLAALDH1A1TSHRHSD17B10
SCHEMBL7358861 0.86 LMNA (0.60) ALDH1A1HSD17B10USP2LMNAPOLB
SCHEMBL2517602 0.84 ALDH1A1 (0.67) AGTR1ALDH1A1TSHRTDP1MAPT
SCHEMBL11148867 0.84 TDP1 (0.66) AGTR1GLAALDH1A1TDP1KMT2A
SCHEMBL10141350 0.83 GLA (0.56) AGTR1GLAALDH1A1TDP1KMT2A
SCHEMBL1422197 0.82 USP2 (0.65) GLAALDH1A1TDP1KMT2AMAPT
SCHEMBL2517123 0.80 MEN1 (0.62) ALDH1A1TDP1KMT2AMAPTMEN1
SCHEMBL3000302 0.79 USP2 (0.59) ALDH1A1TDP1KMT2AMAPTMEN1
SCHEMBL9436741 0.78 GLA (1.00) GLAALDH1A1TDP1KMT2AMAPT
SCHEMBL5453322 0.77 MEN1 (0.58) ALDH1A1TSHRTDP1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402327-B1 Acetamide compounds as glucokinase activators, their process and medicinal applications IMPETIS BIOSCIENCES LTD (IN) 2018-03-07 EP disclosed
EP-2402327-B1 Acetamide compounds as glucokinase activators, their process and medicinal applications IMPETIS BIOSCIENCES LTD (IN) 2018-03-07 EP disclosed
EP-2402327-A1 Acetamide compounds as glucokinase activators, their process and medicinal applications Advinus Therapeutics Private Limited (IN) 2012-01-04 EP disclosed
EP-2402327-A1 Acetamide compounds as glucokinase activators, their process and medicinal applications Advinus Therapeutics Private Limited (IN) 2012-01-04 EP disclosed