SCHEMBL18488113

SCHEMBL18488113

CC(C)c1cc(C=N)ccc1F

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.33
SLC9A1 P19634 1/20 0.32
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18488343 0.80 TYR (0.47)
SCHEMBL29956336 0.80 TYR (0.47)
SCHEMBL18488056 0.80 ALDH1A1 (0.39) NFE2L2SLC9A1PDE2A
SCHEMBL23718577 0.78 CNR2 (0.41) NFE2L2
SCHEMBL8345423 0.73 NFE2L2 (0.50) NFE2L2
SCHEMBL31079293 0.72 GABRA1 (0.46) SLC9A1
SCHEMBL13088831 0.72 GABRA1 (0.44) NFE2L2
SCHEMBL12261433 0.72 GABRA1 (0.46) SLC9A1
SCHEMBL20738711 0.72 GABRA1 (0.39) SLC9A1PDE2A
SCHEMBL18493885 0.72 RPS6KA3 (0.30) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023905-A1 HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF TNF ALPHA BRISTOL-MYERS SQUIBB COMPANY (US) 2017-02-09 WO disclosed